qFit-ligand reveals widespread conformational heterogeneity of drug-like molecules in X-ray electron density maps

By Gydo C. P. Van Zundert, Brandi M. Hudson, Saulo H. P. De Oliveira, Daniel A. Keedy, Rasmus Fonseca, Amelie Heliou, Pooja Suresh, Kenneth Borrelli, Tyler Day, James Fraser1, Henry Van Den Bedem

1. University of California-San Francisco

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journal-article

Author

Gydo C. P. van Zundert and Brandi M. Hudson and Saulo H. P. de Oliveira and Daniel A. Keedy and Rasmus Fonseca and Amelie Heliou and Pooja Suresh and Kenneth Borrelli and Tyler Day and James S. Fraser and Henry van den Bedem

Citation

Van Zundert, G. et al., 2018. qFit-ligand reveals widespread conformational heterogeneity of drug-like molecules in X-ray electron density maps. Journal of Medicinal Chemistry. Available at: http://dx.doi.org/10.1021/acs.jmedchem.8b01292.

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